Empesertib (BAY 1161909)

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

Empesertib (BAY 1161909) 是一种有效的 Mps1 抑制剂，IC50 < 1 nM。

BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM. BAY 1161909 also shows anti-tumor effect, suppressing the proliferation of Hela cells, with an IC50 of < 400 nM.(In Vitro):BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM. BAY 1161909 also shows anti-tumor effect, suppressing the proliferation of Hela cells, with an IC50 of < 400 nM.

BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM. BAY 1161909 also shows anti-tumor effect, suppressing the proliferation of Hela cells, with an IC50 of < 400 nM.

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BAY 1161909

Cell Cycle/DNA Damage

Mps1/TTK

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1443763-60-7

559.61

C??H??FN?O?S

>98% (HPLC)

DMSO : ≥ 35 mg/mL (62.54 mM) H2O : < 0.1 mg/mL (insoluble)

FC1=CC=C([C@@H](C)C(NC2=CC=C(C3=CN4N=C(NC5=CC=C(S(C)(=O)=O)C=C5OC)N=C4C=C3)C=C2)=O)C=C1

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(-20℃)

With Ice Pack

≥ 2 years